平安! 发表于 2011-11-9 19:57 $ P7 i1 G6 Q8 ?0 O
Pazopanib (100 mg/kg/day free base equivalent)
' ^; x- M& P- K) d5 K 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。3 b$ o! P/ W/ |# f, N7 z
搜索了一下,原料一大堆。& w% G: |, L2 R, @1 d/ _# Q2 |
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对不起!100mg/kg是用于移植瘤的,我弄错了。; O$ F& K6 y' \9 }
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以下是正版说明书的推荐用量。
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--------------------- DOSAGE AND ADMINISTRATION ----------------9 [5 e8 I5 }$ J4 m3 c
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) " f9 ~" z+ g8 G1 C* @
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) ! W; [! v! D. I: d- N9 ?/ {" j
---------------------DOSAGE FORMS AND STRENGTHS --------------
$ H+ E2 L/ E. @; C200 mg tablets. (3)
' K" j u: ?4 C) {5 @& l2 E-------------------------------CONTRAINDICATIONS------------------------ |