平安! 发表于 2011-11-9 19:57
! X4 h3 E! V& u9 A( BPazopanib (100 mg/kg/day free base equivalent) ; k/ j- e4 e4 D! G% z$ n& w
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
/ i& G8 i7 I; R% U搜索了一下,原料一大堆。
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对不起!100mg/kg是用于移植瘤的,我弄错了。2 Y5 K* F% R3 N- ^2 F7 L k& D
7 O. y8 ?' E* c" y7 u% s& D/ J以下是正版说明书的推荐用量。" f! v7 I. F/ ^2 n# j$ G% i2 v
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--------------------- DOSAGE AND ADMINISTRATION ----------------
: x2 Q* b* H$ N* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
1 c0 @) z P7 O/ t. F* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
8 y/ X4 \& h8 a" C! n: _---------------------DOSAGE FORMS AND STRENGTHS --------------1 V2 x& c4 X# I+ h+ ^) \* G9 W
200 mg tablets. (3)
) D& b, y: L9 b-------------------------------CONTRAINDICATIONS------------------------ |